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Herbal Extract

Epimedium brevicornum Extract (Leaf) - 10% Icariin

Also known as: Horny Goat Weed, Epimedium, Yin Yang Huo, Icariin

B
Evidence

A traditional Chinese herb extract standardized to 10% icariin, a prenylated flavonol compound used for sexual function and vascular health. Icariin acts as a phosphodiesterase-5 (PDE-5) inhibitor.

Primary uses

  • Sexual function and erectile quality
  • Vascular endothelial function
  • Bone health
  • Energy and stamina

How it works

  • PDE-5 inhibition (similar to pharmaceutical ED drugs)
  • Nitric oxide pathway enhancement
  • Improved blood flow
  • Anti-inflammatory effects

Dosage

Typical range
500-1000 mg daily of 10% icariin extract (providing ~50-100 mg icariin)
Timing
Typically taken 30-60 minutes before sexual activity, or daily for chronic use
With food
May take with or without food; fatty meals may enhance absorption
Duration
Acute effects noted within 1-2 hours; chronic benefits develop over 2-4 weeks of daily use
Special populations
Caution in individuals taking nitrates or other ED medications; monitor blood pressure

Forms

  • Extract· 70/100
  • Capsule· 70/100

Safety

Common side effects

  • Flushing
  • Headache
  • Mild digestive upset
  • Dizziness

Contraindications

  • Concurrent use with nitrates or phosphodiesterase inhibitors (sildenafil, etc.)
  • Uncontrolled hypertension
  • Recent cardiac events
  • Severe liver or kidney disease

Evidence notes

In vivo and clinical studies support PDE-5 inhibition and erectile function improvement; human RCT data is moderate but emerging. 10% icariin is a meaningful standardization level.

Grade B: Some human trials support key claims; further confirmation needed.

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Medical disclaimer. This page is educational and does not replace advice from a qualified healthcare provider.