Mineral
Magnesium Bisglycinate Chelate
Also known as: Magnesium bisglycinate, Magnesium glycinate, Chelated magnesium, Mg bisglycinate
Magnesium bisglycinate is a highly absorbable form of magnesium bound to the amino acid glycine, which enhances intestinal absorption and reduces GI side effects compared to inorganic forms. Strong evidence supports magnesium supplementation for muscle function, sleep quality, stress management, and cardiovascular health.
Primary uses
- Sleep quality and insomnia support
- Muscle relaxation and cramping
- Stress and anxiety management
- Cardiovascular and bone health
- Energy metabolism support
How it works
- Cofactor for 300+ enzymatic reactions including ATP production and protein synthesis
- Regulates neurotransmitter release and nerve function
- Modulates calcium signaling in muscle contraction
- Supports GABA receptors for relaxation and sleep
- Enhances intestinal absorption via glycine carrier when chelated
Dosage
- Typical range
- 200-400 mg elemental magnesium daily
- Timing
- Evening dose recommended for sleep support; can be split morning and evening
- With food
- Can be taken with or without food; bisglycinate form generally well-tolerated either way
- Duration
- Safe for long-term daily use; benefits for sleep typically seen within 2-4 weeks of consistent use
- Special populations
- Pregnant/nursing women should not exceed 350 mg/day; those with kidney disease should consult healthcare provider before supplementing
Forms
- Capsule· 70/100
- Tablet· 70/100
- Powder· 70/100
- Liquid· 70/100
Safety
Common side effects
- Minimal GI distress (advantage over magnesium oxide)
- Loose stools at very high doses (>600 mg/day)
- Rare: drowsiness or headache in sensitive individuals
Contraindications
- Severe kidney disease or renal failure
- Myasthenia gravis
- Heart block or cardiac arrhythmias (high doses)
- Simultaneous use with certain antibiotics (theoretical concern)
Evidence notes
Magnesium supplementation has extensive RCT evidence for multiple health outcomes. The bisglycinate form specifically shows superior absorption and reduced GI distress compared to magnesium oxide; clinical evidence supports improved sleep and muscle function with this chelated form.
Grade A: Multiple well-designed human trials support the main claims.
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